| Date | Insider | Shares | Transaction | Value* |
| 19-Nov-08 | ZAKRZEWSKI JOSEPH S Director | 772,327 | Purchase at $0 per share. | N/A |
| 30-Sep-08 | ZAKRZEWSKI JOSEPH S Director | 125,000 | Purchase at $0.04 per share. | $5,000 |
| 15-Sep-08 | ZAKRZEWSKI JOSEPH S Director | 16,500 | Purchase at $0.04 per share. | $660 |
| 12-Sep-08 | ZAKRZEWSKI JOSEPH S Director | 10,000 | Purchase at $0.04 per share. | $400 |
| 9-Sep-08 | ZAKRZEWSKI JOSEPH S Director | 1,330 | Purchase at $0.04 per share. | $53 |
| 8-Sep-08 | ZAKRZEWSKI JOSEPH S Director | 51,500 | Purchase at $0.04 per share. | $2,060 |
| 5-Sep-08 | ZAKRZEWSKI JOSEPH S Director | 7,051 | Purchase at $0.04 per share. | $282 |
| 27-Aug-08 | ZAKRZEWSKI JOSEPH S Director | 200,000 | Purchase at $0.04 per share. | $8,000 |
| 16-Jul-08 | ZAKRZEWSKI JOSEPH S Director | 10,495 | Purchase at $0.04 per share. | $419 |
| 30-Jun-08 | ZAKRZEWSKI JOSEPH S Director | 75,826 | Purchase at $0.04 per share. | $3,033 |
| 27-Jun-08 | ZAKRZEWSKI JOSEPH S Director | 1,000 | Purchase at $0.04 per share. | $40 |
| 3-Apr-08 | DOV PHARMACEUTICAL INC Director | 100,000 | Purchase at $0.05 per share. | $5,000 |
| 9-Jan-08 | DOV PHARMACEUTICAL INC Director | 13,800 | Purchase at $0.07 per share. | $966 |
| 7-Sep-07 | DOV PHARMACEUTICAL INC Director | 25,000 | Purchase at $0.20 per share. | $5,000 |
| 18-Jun-07 | UBS AG Other | 2,500,000 | Disposition (Non Open Market) | N/A |
| 13-Jun-07 | UBS AG Beneficial Owner (10% or more) | 12,249,875 | Statement of Ownership | N/A |
| 11-Jun-07 | POLYGON GLOBAL OPPORTUNITIES MASTER FUND Beneficial Owner (10% or more) | 12,225,672 | Acquisition (Non Open Market) | N/A |
| 11-Jun-07 | HIGHBRIDGE CAPITAL MANAGEMENT LLC Beneficial Owner (10% or more) | 13,295,418 | Acquisition (Non Open Market) | N/A |